Cholesterol 24-hydroxylase-IN-2

Names

[ CAS No. ]:
1613481-52-9

[ Name ]:
Cholesterol 24-hydroxylase-IN-2

Biological Activity

[Description]:

Cholesterol 24-hydroxylase-IN-2 is an inhibitor of cholesterol 24-hydroxylase (CH24H or CYP46A1), with the IC50 of 5.4 nM. Cholesterol 24-hydroxylase-IN-2 can be used in imaging of cholesterol 24-hydroxylase in mammals[1].

[Related Catalog]:

Signaling Pathways >> Metabolic Enzyme/Protease >> Cytochrome P450
Research Areas >> Others

[References]

[1]. Koike Tatsuki, et al. Preparation of arylpiperidines and arylpiperazines as radiolabeled compounds for use in imaging of cholesterol 24-hydroxylase. World Intellectual Property Organization, WO2015190613 A1 2015-12-17

Chemical & Physical Properties

[ Molecular Formula ]:
C20H23FN4O

[ Molecular Weight ]:
354.42

Related Compounds

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