SC-51089

Names

[ Name ]:
SC-51089

[Synonym ]:
8-chloro-N'-[3-(pyridin-4-yl)propanoyl]dibenzo[b,f][1,4]oxazepine-10(11H)-carbohydrazide
Dibenz[b,f][1,4]oxazepine-10(11H)-carboxylic acid, 8-chloro-, 2-[1-oxo-3-(4-pyridinyl)propyl]hydrazide
8-Chloro-N'-[3-(4-pyridinyl)propanoyl]dibenzo[b,f][1,4]oxazepine-10(11H)-carbohydrazide

Biological Activity

[Description]:

SC-51089 is a selective antagonist of EP1 receptor with analgesic activity in vivo[1].

[Related Catalog]:

Signaling Pathways >> GPCR/G Protein >> Prostaglandin Receptor

Research Areas >> Neurological Disease

[Target]

EP1 Receptor

[References]

[1]. Malmberg AB, et al. Antinociceptive effect of spinally delivered prostaglandin E receptor antagonists in the formalin test on the rat. Neurosci Lett. 1994 May 23;173(1-2):193-6.

Chemical & Physical Properties

[ Density]:
1.4±0.1 g/cm3

[ Boiling Point ]:
633ºC at 760 mmHg

[ Molecular Formula ]:
C₂₂H₁₉ClN₄O₃

[ Molecular Weight ]:
422.864

[ Flash Point ]:
336.6ºC

[ Exact Mass ]:
422.114563

[ PSA ]:
83.56000

[ LogP ]:
2.90

[ Vapour Pressure ]:
2.84E-16mmHg at 25°C

[ Index of Refraction ]:
1.641

Related Compounds

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