PDE5-IN-6c
Names
[ CAS No. ]:
1448419-13-3
[ Name ]:
PDE5-IN-6c
Biological Activity
[Description]:
A novel potent, selective PDE5 inhibitor with IC50 of 0.056 nM for PDE5A1; displays >500-fold selectivity over PDE6; exhibits good efficacy in mouse model of Alzheimer's disease.
[References]
References 1. Fiorito J, et al. J Med Chem. 2017 Nov 9;60(21):8858-8875. View Related Products by Target Phosphodiesterase (PDE)
Chemical & Physical Properties
[ Molecular Formula ]:
C23H21ClN4O2
[ Molecular Weight ]:
420.897