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LY2880070

Names

[ CAS No. ]:
1375637-35-6

[ Name ]:
LY2880070

Biological Activity

[Description]:

LY2880070 is an orally active CHK1 inhibitor. LY2880070 can be used as an anticancer agent for combination with DNA damaging agents[1].

[Related Catalog]:

Research Areas >> Cancer
Signaling Pathways >> Cell Cycle/DNA Damage >> Checkpoint Kinase (Chk)

[Target]

1375637-35-6


[References]

[1]. Quincy S, et al. A phase Ib study of oral Chk1 inhibitor LY2880070 in combination with gemcitabine in patients with advanced or metastatic cancer. Journal of Clinical Oncology 2020 38:15_suppl, 3581.

Chemical & Physical Properties

[ Molecular Formula ]:
C19H23N7O2

[ Molecular Weight ]:
381.43