TAK1-IN-1

Names

[ Name ]:
TAK1-IN-1

Biological Activity

[Description]:

TAK1-IN-1 is a potent, selective, Type I (ATP-competitive, DFG-in) TAK1 inhibitor with Kd of 59 nM, a thienopyrimidine scaffold that serves as a good starting point for medicinal chemistry.

[References]

References 1. Miura T, et al. Bioorg Med Chem Lett. 2017 Feb 15;27(4):1031-1036. View Related Products by Target TAK1

Chemical & Physical Properties

[ Molecular Formula ]:
C₁₇H₁₂N₄O₂S

[ Molecular Weight ]:
336.369

Related Compounds

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