PF-05150122

Names

[ Name ]:
PF-05150122

Biological Activity

[Description]:

PF-05150122 is a potent, state-dependent, subtype selective Nav1.7 inhibitor with IC50 of 21 nM, no significant activity against Nav1.5. Pain Phase 1 Discontinued

[References]

References 1. Swain NA, et al. J Med Chem. 2017 Aug 24;60(16):7029-7042. 2. Jones HM, et al. Clin Pharmacokinet. 2016 Jul;55(7):875-87. View Related Products by Target Sodium Channel Pain

Chemical & Physical Properties

[ Molecular Formula ]:
C₁₉H₁₀ClF₄N₅O₃S₂

[ Molecular Weight ]:
531.885

Related Compounds

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