SW-106

Names

[ Name ]:
SW-106

Biological Activity

[Description]:

A potent, selective, competitive PTH/PTH-related peptide receptor (PPR) antagonist with IC50 of 0.99 uM; displays higher affinity for the PPR relative to the other GPCRs; specificly blocks PTH-initiated cAMP accumulation.

[References]

References 1. Carter PH, et al. Proc Natl Acad Sci U S A. 2007 Apr 17;104(16):6846-51. 2. Carter PH, et al. Mol Endocrinol. 2015 Feb;29(2):307-21. View Related Products by Target PTH Receptor

Chemical & Physical Properties

[ Molecular Formula ]:
C₁₇H₁₆F₅NO₂

[ Molecular Weight ]:
361.312

Related Compounds

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