The Journal of organic chemistry

Synthesis of acridines by the [4+ 2] annulation of arynes and 2-aminoaryl ketones

DC Rogness, RC Larock

Index: Ferencz, Laszlo; Farcasan, Valer; Silberg, Ioan A. Revue Roumaine de Chimie, 2003 , vol. 48, # 10 p. 801 - 811

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Citation Number: 56

Abstract

... a To a sealed 6 dram vial containing 2-aminoacetophenone, the benzyne precursor, a stir bar, and half the total volume of solvent was added CsF, followed by the remainder of the solvent. The reaction was sealed and allowed to stir for a given time before brine (10 mL) was ...

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