Discovery of orally active carboxylic acid derivatives of 2-phenyl-5-trifluoromethyloxazole-4-carboxamide as potent diacylglycerol acyltransferase-1 inhibitors for the …

Y Qian, SJ Wertheimer, M Ahmad…

Index: Journal of Medicinal Chemistry, , vol. 54, # 7 p. 2433 - 2446

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Citation Number: 27

Abstract

... Journal of Medicinal Chemistry. ... Department of Discovery Chemistry, ‡ Non-Clinical Drug Safety, § Metabolism and Pharmacokinetics, ∥ Discovery Technologies, and ⊥ Metabolic and Vascular Diseases, Hoffmann-La Roche Inc., 340 Kingsland Street, Nutley, New Jersey ...

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