Facile synthesis of new substituted aryl and heteroarylflavones by thermal and microwave assisted Suzuki-Miyaura coupling reaction

V Joshi, J Govind Hatim

Index: Joshi, Vidya; Govind Hatim, Jaywant Indian Journal of Chemistry - Section B Organic and Medicinal Chemistry, 2012 , vol. 51, # 7 p. 1002 - 1010

Full Text: HTML

Citation Number: 0

Abstract

Abstract: Microwave assisted Suzuki-Miyaura coupling of 4'-bromoflavone 5 with substituted aryl and heteroarylboronic acids 6a-m gives high yields of aryl and heteroarylflavones 7a-m. Couplings have been carried out by three methods i) conventional heating with Pd (OCOCH 3) 2 catalyst, in solvent DMF (N, N-dimethylformamide) and base, aqueous Na 2 CO 3 (2N) for 6-12 hr, at 110 C, yield 30-70%, ii) conventional heating with Pd [(C 6 H 5) 3 P] 4 ...

Related Articles:

JSCS Vol 7 8, No. 7

[Kulkarni, Pramod S.; Kondhare, Dasharath D.; Varala, Ravi; Zubaidha, Pudukulathan K. Journal of the Serbian Chemical Society, 2013 , vol. 78, # 7 p. 909 - 916]

A novel route to synthesis of flavones from salicylaldehyde and acetophenone derivatives

[Sashidhara, Koneni V.; Kumar, Manoj; Kumar, Abdhesh Tetrahedron Letters, 2012 , vol. 53, # 18 p. 2355 - 2359]

Microwave enhanced palladium catalysed coupling reactions: a diversity-oriented synthesis approach to functionalised flavones

[Fitzmaurice, Richard J.; Etheridge, Zac C.; Jumel, Emelie; Woolfson, Derek N.; Caddick, Stephen Chemical Communications, 2006 , # 46 p. 4814 - 4816]

Pd–carbene catalyzed carbonylation reactions of aryl iodides

[Xue, Liqin; Shi, Lijun; Han, Yuan; Xia, Chungu; Huynh, Han Vinh; Li, Fuwei Dalton Transactions, 2011 , vol. 40, # 29 p. 7632 - 7638]

One-step conversion of flavanones into isoflavones: a new facile biomimetic synthesis of isoflavones

[Tetrahedron Letters, , vol. 31, # 50 p. 7355 - 7356]

More Articles...