Synthesis of 5-arylpyrrolo [1, 2-c] pyrimidin-1 (2 H)-ones

M Álvarez, D Fernández, JA Joule

Index: Alvarez, Mercedes; Fernandez, David; Joule, John A. Journal of the Chemical Society. Perkin Transactions 1, 2002 , # 4 p. 471 - 475

Full Text: HTML

Citation Number: 0

Abstract

In a previous paper 3 we described the preparation of simplified structural analogues of the variolins, lacking the pyrimidine ring, using the Stille reaction between 3-trimethylstannyl-7-azaindoles and aromatic halides. None of the 3-aryl-7-azaindoles thus prepared showed activities ...