4-(Aminoacylamido)-s-hydrindacenes and related compounds: Synthesis and pharmacological screening

…, J Holubek, M Bartošová, M Protiva

Index: Vejdelek; Holubek; Bartosova; Protiva Collection of Czechoslovak Chemical Communications, 1982 , vol. 47, # 12 p. 3297 - 3305

Full Text: HTML

Citation Number: 2

Abstract

Abstract Chloracylamido derivatives IIIa-Va were obtained by acylation of 4-amino-s- hydrindacene with chloroacetyl chloride, 2-chloropropionyl chloride and 3-chloropropionyl chloride; their reactions with excessive diethylamine, pyrrolidine, piperidine and morpholine afforded the title compounds IIIbcde-Vbcde. A reaction of 4-amino-s-hydrindacene with benzoyl isothiocyanate gave 1-benzoyl-3-(s-hydrindacen-4-yl) thiourea (VI) whose mild ...

Related Articles:

Novel synthesis of 1-(1, 2, 3, 5, 6, 7-hexahydro-s-indacen-4-yl)-3-[4-(1-hydroxy-1-methyl-ethyl)-furan-2-sulfonyl] urea, an anti-inflammatory agent

[Urban, Frank J.; Jasys, V. John; Raggon, Jeffrey W.; Buzon, Richard A.; Hill, Paul D.; Eggler, James F.; Weaver, John D. Synthetic Communications, 2003 , vol. 33, # 12 p. 2029 - 2043]

4-(Aminoacylamido)-s-hydrindacenes and related compounds: Synthesis and pharmacological screening

[Vejdelek; Bartosova; Protiva Collection of Czechoslovak Chemical Communications, 1977 , vol. 42, # 6 p. 1992 - 2000]

Difunctional derivatives of syn-dimethanoperhydro-s-hydrindacene

[Birladeanu,L. et al. Journal of Organic Chemistry, 1977 , vol. 42, # 20 p. 3260 - 3264]

Novel synthesis of 1-(1, 2, 3, 5, 6, 7-hexahydro-s-indacen-4-yl)-3-[4-(1-hydroxy-1-methyl-ethyl)-furan-2-sulfonyl] urea, an anti-inflammatory agent

[Urban, Frank J.; Jasys, V. John; Raggon, Jeffrey W.; Buzon, Richard A.; Hill, Paul D.; Eggler, James F.; Weaver, John D. Synthetic Communications, 2003 , vol. 33, # 12 p. 2029 - 2043]

Novel synthesis of 1-(1, 2, 3, 5, 6, 7-hexahydro-s-indacen-4-yl)-3-[4-(1-hydroxy-1-methyl-ethyl)-furan-2-sulfonyl] urea, an anti-inflammatory agent

[Urban, Frank J.; Jasys, V. John; Raggon, Jeffrey W.; Buzon, Richard A.; Hill, Paul D.; Eggler, James F.; Weaver, John D. Synthetic Communications, 2003 , vol. 33, # 12 p. 2029 - 2043]

More Articles...