Major effect of pyrrolic N-benzylation in norbinaltorphimine, the selective κ-opioid receptor antagonist

C Chauvignac, CN Miller, SK Srivastava…

Index: Journal of Medicinal Chemistry, , vol. 48, # 5 p. 1676 - 1679

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Citation Number: 5

Abstract

... Journal of Medicinal Chemistry. ... analogues, plus the further evaluation of 1b in vivo. figure. Chemistry. Two complimentary methods were utilized for the synthesis of BnorBNI (1b). In the first, the reported method for the ...