Organic letters

Stereoselective synthesis of a dioxa-bicyclo [3.2. 1] octane SGLT2 inhibitor

V Mascitti, C Préville

Index: Organic Letters, , vol. 12, # 13 p. 2940 - 2943

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Citation Number: 13

Abstract

... Volume: Page: Digital Object Identifier (DOI). ... Organic Letters. ... When 8 was stirred at 23 °C in a mixture of TFA/H 2 O (9/1 vol.) under air, deprotection/cyclization occurred to cleanly produce 1 as a single isomer in 77% yield. ...