Tetrahedron Letters

Optically active N-hydroxytartrimides for enantioselective peptide synthesis

T Teramoto, M Deguchi, T Kurosaki, M Okawara

Index: Teramoto, Takero; Deguchi, Mikito; Kurosaki, Toshikazu; Okawara, Makoto Tetrahedron Letters, 1981 , vol. 22, p. 1109 - 1112

Full Text: HTML

Citation Number: 22

Abstract

Abstract Preparations of optically active N-hydroxytartrimides were achieved. 1, 3, 4- Trihydroxysuccinimide ester of ZL-alanine and 1-hydroxy-3, 4-diacetoxysuccinimide ester of ZD-alanine were allowed to react with D, L-alaninate to produce LL form and DD form of Z- Ala-Ala-OEt respectively (optical yield 100%).

Related Articles:

Small peptides as modular catalysts for the direct asymmetric aldol reaction: ancient peptides with aldolase enzyme activity

[Zou, Weibiao; Ibrahem, Ismail; Dziedzic, Pawel; Sunden, Henrik; Cordova, Armando Chemical Communications, 2005 , # 39 p. 4946 - 4948]

Small peptides as modular catalysts for the direct asymmetric aldol reaction: ancient peptides with aldolase enzyme activity

[Zou, Weibiao; Ibrahem, Ismail; Dziedzic, Pawel; Sunden, Henrik; Cordova, Armando Chemical Communications, 2005 , # 39 p. 4946 - 4948]

1, 1'-Bis [6-(trifluoromethyl) benzotriazolyl] oxalate (BTBO): a new reactive coupling reagent for the synthesis of dipeptides, esters, and thio esters

[Takeda, Kazuyoshi; Tsuboyama, Kanoko; Yamaguchi, Keiko; Ogura, Haruo Journal of Organic Chemistry, 1985 , vol. 50, # 2 p. 273 - 275]

Kinetics of the alkaline hydrolysis of several N-benzyloxycarbonyldipeptide methyl and ethyl esters

[Hoogwater, D. A.; Peereboom, M. Tetrahedron, 1990 , vol. 46, # 15 p. 5325 - 5332]

Kinetics of the alkaline hydrolysis of several N-benzyloxycarbonyldipeptide methyl and ethyl esters

[Hoogwater, D. A.; Peereboom, M. Tetrahedron, 1990 , vol. 46, # 15 p. 5325 - 5332]

More Articles...