Tetrahedron

Pyridinium N-(2′-Azinyl) Aminides: Regioselective Synthesis of 2-Alkylaminoazines

…, JL Garcıa-Navıo, ML Izquierdo, J Alvarez-Builla

Index: Martinez-Barrasa, Valentin; Delgado, Francisca; Burgos, Carolina; Luis Garcia-Navio; Luisa Izquierdo; Alvarez-Builla, Julio Tetrahedron, 2000 , vol. 56, # 16 p. 2481 - 2490

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Citation Number: 34

Abstract

Download PDF Opens in a new window. Article suggestions will be shown in a dialog on return to ScienceDirect. ... Please enable JavaScript to use all the features on this page. ... The regioselective alkylation of pyridinium-N-(2′-azinil)aminides with alkyl halides under mild conditions is described. The alkylation, combined with a reduction of the N–N bond, allows an easy preparation of 2-alkylaminoazines. ... Generally, regioselectivity of the substitution reaction can be ...

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