A mild method for formylating amino esters without using any formylating agent
T Giard, D Bénard, JC Plaquevent
Index: Giard, Thierry; Benard, Didier; Plaquevent, Jean-Christophe Synthesis, 1998 , # 3 p. 297 - 300
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Citation Number: 9
Abstract
Abstract: A simple and mild method for the N-formylation of _-amino esters is described via an intermediate oxaziridine. This procedure avoids the necessity of specific formylating agents and yields the N-formyl species in high yield and without racemization. Key words: formylation, amino esters, oxaziridines, imines, Möhr's salt
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