An Integrated Chemo-enzymatic Route for Preparation of β-Thymidine, a Key Intermediate in the Preparation of Antiretrovirals

GER Gordon, ML Bode, DF Visser…

Index: Organic Process Research and Development, , vol. 15, # 1 p. 258 - 265

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Abstract

... Organic Process Research & Development. ... The general process followed from 5-MU to DABT was first described by Mansuri et al.(8) This reaction proceeds via an ... in that a saturated brine wash, instead of a water wash, was applied to minimise transfer of organics into the ...

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