… ) of Bis (aroylmethyl) Sulfides (= 1, 1′??[Thiobis (methylene)] bis [arylmethanone] Bis (2??phenylhydrazones)): Synthesis of 3??Aroylindoles (= Aryl (1H??indol??3??yl) …
N Paul, S Muthusubramanian
Index: Paul, Nidhin; Muthusubramanian, Shanmugam Helvetica Chimica Acta, 2013 , vol. 96, # 3 p. 452 - 457
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Abstract
Abstract The bis (phenylhydrazone) of substituted diphenacyl sulfides (= 1, 1′-[thiobis (methylene)] bis [arylmethanone] bis (2-phenylhydrazones)) 1 underwent a tandem sequence of reactions upon treatment with Vilsmeier reagent, ultimately yielding 3- aroylindoles (= aryl (1H-indol-3-yl) methanones) 3 (Scheme 1 and Table 1). The reaction seems to be product selective depending upon the reaction temperature.
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