Chinese Chemical Letters

Synthesis of 3-acylindoles via decarboxylative cross-coupling reaction of free (NH) indoles with α-oxocarboxylic acids

LJ Gu, JY Liu, LZ Zhang, Y Xiong, R Wang

Index: Gu, Li-Jun; Liu, Ji-Yan; Zhang, Li-Zhu; Xiong, Yong; Wang, Rui Chinese Chemical Letters, 2014 , vol. 25, # 1 p. 90 - 92

Full Text: HTML

Citation Number: 19

Abstract

A convenient and general method for acylation of free (N H) indoles via palladium-catalyzed decarboxylative cross-coupling reaction was developed. This process provided a useful method for the preparation of diverse 3-acylindoles in high yields utilizing a reaction with readily accessible reactants under mild conditions. ... A convenient method for the preparation of 3-acylindoles via palladium-catalyzed decarboxylative cross-coupling reaction of free (N H) indoles with ...

Related Articles:

Normal electron demand Diels–Alder cycloaddition of indoles to 2, 3-dimethyl-1, 3-butadiene

[De La Fuente, M. Carmen; Dominguez, Domingo Tetrahedron, 2011 , vol. 67, # 22 p. 3997 - 4001]

Normal electron demand Diels–Alder cycloaddition of indoles to 2, 3-dimethyl-1, 3-butadiene

[De La Fuente, M. Carmen; Dominguez, Domingo Tetrahedron, 2011 , vol. 67, # 22 p. 3997 - 4001]

A systematic study of two complementary protocols allowing the general, mild and efficient deprotection of N-pivaloylindoles

[Ruiz, Miriam; Sanchez, J. Domingo; Lopez-Alvarado, Pilar; Menendez, J. Carlos Tetrahedron, 2012 , vol. 68, # 2 p. 705 - 710]

Meridianin G and its analogs as antimalarial agents

[Bharate, Sandip B.; Yadav, Rammohan R.; Khan, Shabana I.; Tekwani, Babu L.; Jacob, Melissa R.; Khan, Ikhlas A.; Vishwakarma, Ram A. MedChemComm, 2013 , vol. 4, # 6 p. 1042 - 1048]

A convenient synthesis of 3-acylindoles via Friedel Crafts acylation of 1-(phenylsulfonyl) indole. A new route to pyridocarbazole-5, 11-quinones and ellipticine

[Ketcha, Daniel M.; Gribble, Gordon W. Journal of Organic Chemistry, 1985 , vol. 50, # 26 p. 5451 - 5457]

More Articles...