β-Naphthoflavone analogs as potent and soluble aryl hydrocarbon receptor agonists: Improvement of solubility by disruption of molecular planarity
Y Fujita, M Yonehara, M Tetsuhashi…
Index: Bioorganic and Medicinal Chemistry, , vol. 18, # 3 p. 1194 - 1203
Full Text: HTML
Citation Number: 27
Abstract
... Please enable JavaScript to use all the features on this page. Bioorganic & Medicinal Chemistry. Volume 18, Issue 3, 1 February 2010, Pages 1194–1203. ... Here, we describe chemical modification of an AhR agonist, β-naphthoflavone, focusing on planarity-disruption. ...
Related Articles:
Synthesis and biological evaluation of flavones and benzoflavones as inhibitors of BCRP/ABCG2
[Juvale, Kapil; Stefan, Katja; Wiese, Michael European Journal of Medicinal Chemistry, 2013 , vol. 67, p. 115 - 126]
[Fujita, Yuji; Yonehara, Mitsuhiro; Tetsuhashi, Masashi; Noguchi-Yachide, Tomomi; Hashimoto, Yuichi; Ishikawa, Minoru Bioorganic and Medicinal Chemistry, 2010 , vol. 18, # 3 p. 1194 - 1203]
[Garg, S.; Ishar, M. P. S.; Sarin, R.; Gandhi, R. P. Indian Journal of Chemistry, Section B: Organic Chemistry Including Medicinal Chemistry, 1994 , vol. 33, # 12 p. 1123 - 1128]
Synthesis and biological evaluation of flavones and benzoflavones as inhibitors of BCRP/ABCG2
[European Journal of Medicinal Chemistry, , vol. 67, p. 115 - 126]
Synthesis and biological evaluation of flavones and benzoflavones as inhibitors of BCRP/ABCG2
[European Journal of Medicinal Chemistry, , vol. 67, p. 115 - 126]