Exploiting subsite S1 of trypsin-like serine proteases for selectivity: potent and selective inhibitors of urokinase-type plasminogen activator

RL Mackman, BA Katz, JG Breitenbucher…

Index: Imakura; Okimoto; Konishi; Hisazumi; Yamazaki; Kobayashi; Yamashita Chemical and Pharmaceutical Bulletin, 1992 , vol. 40, # 7 p. 1691 - 1696

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Citation Number: 76

Abstract

... Departments of Medicinal Chemistry, Structural Biology, and Preclinical Sciences, Axys Pharmaceuticals Inc., 180 ... Chem. , 2001, 44 (23), pp 3856–3871. DOI: 10.1021/jm010244+. Publication Date (Web): October 6, 2001. Copyright © 2001 American Chemical Society. ...