MedChemComm

2-[18 F] Fluoroethyl tosylate–a versatile tool for building 18 F-based radiotracers for positron emission tomography

T Kniess, M Laube, P Brust, J Steinbach

Index: Bauman; Piel; Hoehnemann; Krauss; Jansen; Solbach; Dannhardt; Roesch Journal of Labelled Compounds and Radiopharmaceuticals, 2011 , vol. 54, # 10 p. 645 - 656

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Abstract

... properties like ethyl and methyl groups and is expected to maintain the pharmacological properties of a lead compound. ... Rösch et al. ... synthesized 18 F-labeled compounds derived from FAUC346 with the methoxy functionality being replaced with a fluoroethoxy bioisostere (Fig. ...

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