Tetrahedron Letters

Microwave-assisted synthesis of 1-aminoalkyl phosphonates under solvent-free conditions

B Kaboudin, R Nazari

Index: Kaboudin, Babak; Nazari, Rahman Tetrahedron Letters, 2001 , vol. 42, # 46 p. 8211 - 8213

Full Text: HTML

Citation Number: 201

Abstract

A simple, efficient and general method has been developed for the synthesis of 1-aminoalkyl phosphonates through a one-pot reaction of aldehydes with amines in the presence of acidic alumina under solvent-free conditions using microwave irradiation. It was also found that acidic alumina supported ammonium formate under solvent-free conditions is capable of the synthesis of 1-aminophosphonates from aldehydes and diethyl phosphite under ...

Related Articles:

Synthesis, physical and biological properties of the phosphorus analogues of phenylalanine and related compounds

[Maier, Ludwig; Diel, Peter J. Phosphorus, Sulfur and Silicon and the Related Elements, 1991 , vol. 57, # 1/2 p. 57 - 64]

Synthesis and antitumor activities of novel rhein α-aminophosphonates conjugates

[Yao, Gui-Yang; Ye, Man-Yi; Huang, Ri-Zhen; Li, Ya-Jun; Pan, Ying-Ming; Xu, Qing; Liao, Zhi-Xin; Wang, Heng-Shan Bioorganic and Medicinal Chemistry Letters, 2014 , vol. 24, # 2 p. 501 - 507]

Synthesis and antitumor activities of novel α-aminophosphonates dehydroabietic acid derivatives

[Huang, Xiao-Chao; Wang, Meng; Pan, Ying-Ming; Tian, Xiao-Yan; Wang, Heng-Shan; Zhang, Ye Bioorganic and Medicinal Chemistry Letters, 2013 , vol. 23, # 19 p. 5283 - 5289]

Synthesis, physical and biological properties of the phosphorus analogues of phenylalanine and related compounds

[Maier, Ludwig; Diel, Peter J. Phosphorus, Sulfur and Silicon and the Related Elements, 1991 , vol. 57, # 1/2 p. 57 - 64]

More Articles...