Synthesis of Benzimidazoles by PIDA??Promoted Direct C (sp2) H Imidation of N??Arylamidines

J Huang, Y He, Y Wang, Q Zhu

Index: Huang, Jinbo; He, Yimiao; Wang, Yong; Zhu, Qiang Chemistry - A European Journal, 2012 , vol. 18, # 44 p. 13964 - 13967

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Citation Number: 54

Abstract

The development of effective methods for the construction of CÀN bonds has received considerable interest of organic chemists because of their ubiquitous existence in pharmaceuticals, agrochemicals, and biologically relevant molecules.[1] Transition-metal- catalyzed amination/amidation/imidation reactions starting from aryl or vinylACHTUNGTRENNUNG (pseudo) halides have been recognized as powerful ...

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