Tyrphostins. II. Heterocyclic and. alpha.-substituted benzylidenemalononitrile tyrphostins as potent inhibitors of EGF receptor and ErbB2/neu tyrosine kinases

A Gazit, N Osherov, I Posner, P Yaish…

Index: Journal of Medicinal Chemistry, , vol. 34, # 6 p. 1896 - 1907

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Citation Number: 254

Abstract

... Journal of Medicinal Chemistry, 1991, Vol. 34, No. 6 1897 Table 11. Structures and Inhibitory and Antiproliferative Activities of Conformationallv Constrained TvrDhostins IC,, p M biochemical data:a biological dahb PolyGAT EGF dependent chemical data no. ...

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