Tetrahedron Letters

Copper-catalysed benzofuran synthesis: developing aryl bromide–alkenyl triflates as general heterocycle precursors

AC Tadd, MR Fielding, MC Willis

Index: Tadd, Andrew C.; Fielding, Mark R.; Willis, Michael C. Tetrahedron Letters, 2007 , vol. 48, # 43 p. 7578 - 7581

Full Text: HTML

Citation Number: 28

Abstract

Download PDF Opens in a new window. Article suggestions will be shown in a dialog on return to ScienceDirect. ... Please enable JavaScript to use all the features on this page. ... A range of conjugated aryl bromide–alkenyl triflates, previously described as indole precursors, are efficiently converted to the corresponding benzofurans when treated with CuI/TMEDA and potassium hydroxide. ... A range of conjugated aryl bromide–alkenyl triflates are efficiently ...

Related Articles:

Palladium-catalysed intramolecular enolate O-arylation and thio-enolate S-arylation: synthesis of benzo [b] furans and benzo [b] thiophenes

[Willis, Michael C.; Taylor, Dawn; Gillmore, Adam T. Tetrahedron, 2006 , vol. 62, # 49 p. 11513 - 11520]

Palladium-catalysed intramolecular enolate O-arylation and thio-enolate S-arylation: synthesis of benzo [b] furans and benzo [b] thiophenes

[Willis, Michael C.; Taylor, Dawn; Gillmore, Adam T. Tetrahedron, 2006 , vol. 62, # 49 p. 11513 - 11520]

Aryne and SNAr reactions of polyhalobenzenes. 6. Synthesis of benzofurans

[Bachelet, Jean-Pierre; Caubere, Paul Journal of Organic Chemistry, 1982 , vol. 47, # 2 p. 234 - 238]

Cascade Palladium??Catalyzed Direct Intramolecular Arylation/Alkene Isomerization Sequences: Synthesis of Indoles and Benzofurans

[Yagoubi, Myriam; Cruz, Ana C. F.; Nichols, Paula L.; Elliott, Richard L.; Willis, Michael C. Angewandte Chemie - International Edition, 2010 , vol. 49, # 43 p. 7958 - 7962]

Dehydrative C–H Alkylation and Alkenylation of Phenols with Alcohols: Expedient Synthesis for Substituted Phenols and Benzofurans

[Lee, Dong-Hwan; Kwon, Ki-Hyeok; Yi, Chae S. Journal of the American Chemical Society, 2012 , vol. 134, # 17 p. 7325 - 7328]

More Articles...