5′-O-Alkylpyridoxamines: Lipophilic Analogues of Pyridoxamine Are Potent Scavengers of 1, 2-Dicarbonyls

V Amarnath, K Amarnath, J Avance…

Index: Zagol-Ikapitte, Irene; Amarnath, Venkataraman; Bala, Manju; Roberts II, L. Jackson; Oates, John A.; Boutaud, Olivier Chemical Research in Toxicology, 2010 , vol. 23, # 1 p. 240 - 250

Full Text: HTML

Citation Number: 3

Abstract

Pyridoxamine (PM) is a prospective drug for the treatment of diabetic complications. In order to make zwitterionic PM more lipophilic and improve its tissue distribution, PM derivatives containing medium length alkyl groups on the hydroxymethyl side chain were prepared. The

Related Articles:

Active core structure of terfestatin A, a new specific inhibitor of auxin signaling

[Hayashi, Ken-ichiro; Yamazoe, Atsushi; Ishibashi, Yuki; Kusaka, Naoyuki; Oono, Yutaka; Nozaki, Hiroshi Bioorganic and Medicinal Chemistry, 2008 , vol. 16, # 9 p. 5331 - 5344]

Design, synthesis and anticancer activities of diaryl urea derivatives bearing N-acylhydrazone moiety

[Zhang, Bei; Zhao, Yanfang; Zhai, Xin; Wang, Lihui; Yang, Jingyu; Tan, Zehui; Gong, Ping Chemical and Pharmaceutical Bulletin, 2012 , vol. 60, # 8 p. 1046 - 1054]

Mild and rapid method for the generation of o-quinone methide intermediates. Synthesis of puupehedione analogues

[Barrero, Alejandro F.; Quilez del Moral, Jose F.; Mar Herrador; Arteaga, Pilar; Cortes, Manuel; Benites, Julio; Rosellon, Antonio Tetrahedron, 2006 , vol. 62, # 25 p. 6012 - 6017]

More Articles...