2-Arylbenzoxazoles as CETP inhibitors: Substitution and modification of the α-alkoxyamide moiety

JA Hunt, S Gonzalez, ML Hammond…

Index: Bioorganic and Medicinal Chemistry Letters, , vol. 20, # 3 p. 1019 - 1022

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Citation Number: 19

Abstract

... Bioorganic & Medicinal Chemistry Letters. ... In this Letter, we describe optimization of the α-aryloxyamide moiety of the screening lead 1, resulting in identification of potent alkyl-substituted analogs such as 3. However, both the α-aryloxyamides and the β-alkyloxyamides ...