Tetrahedron: Asymmetry

The effect of substituents on the chiral solvating properties of (S)-1, 6-dialkylpiperazine-2, 5-diones

Č Malavašič, B Stanovnik, J Wagger, J Svete

Index: Malavasic, Crt; Stanovnik, Branko; Wagger, Jernej; Svete, Jurij Tetrahedron Asymmetry, 2011 , vol. 22, # 12 p. 1364 - 1371

Full Text: HTML

Citation Number: 1

Abstract

The effect of substituents on the chiral solvating properties of 13 different (S)-1, 6- dialkylpiperazine-2, 5-diones (S)-1a–m and five (3S, 6S)-1, 3, 6-trialkyl analogues (S, S)-1n– r was studied by NMR in CDCl3 with methyl (RS)-N-benzoylleucinate (RS)-2a as the model analyte. Most diketopiperazines exhibited typical resolution, ΔΔδRS-20∼ 0.1 ppm. Increased performance was observed with 6-CH2R substituted compounds (S)-1h–j. The ...

Related Articles:

Versatility of cyclooctadiene ligands in iridium chemistry and catalysis

[Cabeza, Javier A.; Cativiela, Carlos; de Villegas, Maria D. Diaz; Oro, Luis A. Journal of the Chemical Society, Perkin Transactions 1: Organic and Bio-Organic Chemistry (1972-1999), 1988 , p. 1881 - 1884]

Use of enantio-, chemo-and regioselectivity of acylase I. Resolution of polycarboxylic acid esters

[Liljeblad, Arto; Aksela, Reijo; Kanerva, Liisa T. Tetrahedron Asymmetry, 2001 , vol. 12, # 14 p. 2059 - 2066]

Asymmetric reactions catalyzed by chiral metal complexes. XXXIII. Efficient asymmetric hydrogenations of (Z)-2-acetamidoacrylic acid derivatives with the cationic …

[Takahashi, Hisashi; Achiwa, Kazuo Chemistry Letters, 1989 , p. 305 - 308]

A general and accurate nmr determination of the enantiomeric purity of α-aminoacids and α-aminoacid derivatives

[Calmes, Monique; Daunis, Jacques; Jacquier, Robert; Verducci, Jean Tetrahedron, 1987 , vol. 43, # 10 p. 2285 - 2292]

Synthesis and incorporation of [3-3H, U-14C]-l-valine into penicillin V using Penicillium chrysogenum

[Wolfe; Bowers; Lowe; Morin Canadian Journal of Chemistry, 1982 , vol. 60, # 3 p. 355 - 361]

More Articles...