Tandem Intramolecular Carbolithiation??Lithium/Zinc Transmetallation and Applications to Carbon− Carbon Bond??Forming Reactions
M Yus, R Ortiz
Index: Yus, Miguel; Ortiz, Rosa European Journal of Organic Chemistry, 2004 , # 18 p. 3833 - 3841
Full Text: HTML
Citation Number: 8
Abstract
Abstract Lithium/zinc transmetallation with the cyclic organolithium intermediate 3 (prepared by intramolecular carbolithiation of the initially formed organolithium 2) gives the corresponding organozinc intermediate 5. Copper-or palladium-promoted SN 2′ reactions between compound 5 and allylic or propargylic halides, as well as arylation, vinylation, benzylation, acylation, and conjugate addition to α, β-unsaturated carbonyl compounds, ...
Related Articles:
Intramolecular carbolithiation promoted by a DTBB-catalysed chlorine–lithium exchange
[Yus, Miguel; Ortiz, Rosa; Huerta, Fernando F. Tetrahedron, 2003 , vol. 59, # 43 p. 8525 - 8542]
Synthesis and evaluation of 4-alkylanilines as mammary tumor inhibiting aromatase inhibitors
[Hartmann; Batzl European Journal of Medicinal Chemistry, 1992 , vol. 27, # 5 p. 537 - 544]
Vanadium-catalyzed cross-coupling reactions of alkyl halides with aryl Grignard reagents
[Yasuda, Shigeo; Yorimitsu, Hideki; Oshima, Koichiro Bulletin of the Chemical Society of Japan, 2008 , vol. 81, # 2 p. 287 - 290]
[Moore,W.M. et al. Journal of the American Chemical Society, 1975 , vol. 97, # 17 p. 4954 - 4960]
[Guennouni; Lhermitte; Cochard; Carboni Tetrahedron, 1995 , vol. 51, # 25 p. 6999 - 7018]