OMDM-5

Modify Date: 2024-01-30 18:10:09

OMDM-5 structure	Common Name	OMDM-5
	CAS Number	616884-66-3	Molecular Weight	432.64
	Density	N/A	Boiling Point	N/A
	Molecular Formula	C₂₆H₄₄N₂O₃	Melting Point	N/A
	MSDS	N/A	Flash Point	N/A

Use of OMDM-5

OMDM-5 is a selective inhibitor of anandamide cellular uptake (ACU), with a Ki of 4.8 μM. OMDM-5 is also a potent vanilloid receptor type 1 (VR1, TRPV1) agonist, with an EC50 of 75 nM, and shows weakly active as cannabinoid receptor type 1 (CB1) ligand (Ki=4.9 μM)[1].

Name	OMDM-5

Description	OMDM-5 is a selective inhibitor of anandamide cellular uptake (ACU), with a Ki of 4.8 μM. OMDM-5 is also a potent vanilloid receptor type 1 (VR1, TRPV1) agonist, with an EC50 of 75 nM, and shows weakly active as cannabinoid receptor type 1 (CB1) ligand (Ki=4.9 μM)[1].
Related Catalog	Signaling Pathways >> Membrane Transporter/Ion Channel >> TRP Channel Research Areas >> Neurological Disease
Target	Ki: 4.8 μM (anandamide cellular uptake), 4.9 μM (CB1), EC50: 75 nM (VR1)[1]
References	[1]. Ortar G, et al. Novel selective and metabolically stable inhibitors of anandamide cellular uptake. Biochem Pharmacol. 2003 May 1;65(9):1473-81.

Molecular Formula	C₂₆H₄₄N₂O₃
Molecular Weight	432.64

OMDM-5

Use of OMDM-5

Names

OMDM-5 Biological Activity

Chemical & Physical Properties