CS-3150
Published date: 2020-01-06 17:06:19
|
Name | Esaxerenone | CAS# | 1632006-28-0 |
|---|---|---|---|---|
| Price | $600.0/100mg $1200.0/250mg $2400.0/1g | Purity | 98.0% | |
| Stocking Period |
3 Day | Stock | In Stock | |
| Product Webpage: | https://www.dcchemicals.com/product_show-DC20999.html | |||
| Detail
Product Information
CS-3150 (Esaxerenone, XL-550) is a highly potent, selective and orally active non-steroidal mineralocorticoid receptor antagonist with IC50 of 9.4 nM; displays >1,000-fold selectivity over other steroid hormone receptors, glucocorticoid receptor, androgen receptor and progesterone receptor; inhibits aldosterone-induced transcriptional activation of human mineralocorticoid receptor with IC50 of 3.7 nM, shows superior potency to that of spironolactone and eplerenone; suppresses aldosterone-induced decrease in urinary Na(+)/K(+) ratio, inhibits blood pressure elevation induced by DOCA/salt-loading in rats. |
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