Synthesis and Neuropeptide Y Y1 Receptor Antagonistic Activity of N, N??Disubstituted ω??Guanidino??and ω??Aminoalkanoic Acid Amides

…, S Dove, G Bernhardt, A Buschauer

Index: Buschauer, Armin Archiv der Pharmazie (Weinheim, Germany), 1989 , vol. 322, p. 165 - 171

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Citation Number: 32

Abstract

Abstract Potent arpromidine-type histamine H 2 receptor agonists such as BU-E-76 (He 90481) were among the first non-peptides reported to display weak neuropeptide Y (NPY) Y 1 receptor antagonist activity. In search of new chemical leads for the development of more