Tetrahedron

Solid-phase synthesis of 4-triphenylphosphoranylidene-4, 5-dihydropyrazol-5-ones, 4-aminocarbonyl-pyrroles, 4-methoxy-1H-pyrazol-5 (2H)-ones and 2-thiazolin-4- …

OA Attanasi, L De Crescentini, P Filippone, F Mantellini…

Index: Attanasi, Orazio A; De Crescentini, Lucia; Filippone, Paolino; Mantellini, Fabio; Tietze, Lutz F Tetrahedron, 2001 , vol. 57, # 27 p. 5855 - 5863

Full Text: HTML

Citation Number: 21

Abstract

Combinatorial synthesis of small organic molecules has evolved rapidly in the last few years to become a new paradigm for contemporary drug discovery. 1 For this reason, increasing attention is currently devoted to this technique. 2 Some of us previously reported the use of modified Merrifield resin in the preparation of polymer-bound β-dicarbonyl derivatives from which some heterocyclic products were obtained. 3 Since 1,2-diaza-1,3-butadienes showed to be useful building ...