Organic letters

Functionalization of Unprotected Uracil Derivatives Using the Halogen-Magnesium Exchange

F Kopp, P Knochel

Index: Organic Letters, , vol. 9, # 9 p. 1639 - 1641

Full Text: HTML

Citation Number: 39

Abstract

... Volume: Page ... Organic Letters. ... 13 More efficiently, the reaction of 7b with benzyl bromide after transmetalation using CuI·2LiCl furnishes the uracil derivative 9 in 57% yield (Scheme 1). The resulting products 8 and 9 are precursors of HEPT (10) and Emivirine (11 ...