Green Chemistry

H 2 O 2-mediated oxidative formation of amides from aromatic amines and 1, 3-diketones as acylation agents via C–C bond cleavage at room temperature in water …

X Sun, M Wang, P Li, X Zhang, L Wang

Index: Sun, Xi; Wang, Min; Li, Pinhua; Zhang, Xiuli; Wang, Lei Green Chemistry, 2013 , vol. 15, # 12 p. 3289 - 3294

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Citation Number: 21

Abstract

The importance and value of amide motifs can be shown from their wide occurrence in natural products, pharmaceuticals, polymers, and biological systems, and their broad applications as versatile building blocks in organic synthesis. 13 As a result, the synthesis of amides is a greatly valuable project and a variety of methods are available for their preparation, such as: the acylation of amines using carboxylic acids or their derivatives; 14 transition-metal-catalyzed ...

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