Tetrahedron letters

A general method for the n-alkylation of thioamides.

AR Katritzky, M Drewniak

Index: Katritzky, Alan R.; Drewniak, Malgorzata Tetrahedron Letters, 1988 , vol. 29, # 15 p. 1755 - 1758

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Citation Number: 45

Abstract

Download full text in PDF Opens in a new window. Article suggestions will be shown in a dialog on return to ScienceDirect. ... Please enable JavaScript to use all the features on this page. ... Thioamides are N-alkylated in a two-step procedure: (i) Reaction with an aldehyde and benzotriazole yields an adduct which is (ii) reduced to the N-alkylthiomide by NaBH 4 . ... AR Katritzky, K. Yannakopoulou, W. Kuzmierkiewicz, JM Aurrecoechea, GJ Palenik, AE Koziol, M. ...

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