Tetrahedron

One-pot synthesis of new aza-and diaza-aminophenanthrenes

…, J Sopková-de Oliveira Santos, S Rault, P Dallemagne

Index: Rochais, Christophe; Yougnia, Rodrigue; Cailly, Thomas; Sopkova-De Oliveira Santos, Jana; Rault, Sylvain; Dallemagne, Patrick Tetrahedron, 2011 , vol. 67, # 32 p. 5806 - 5810

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Citation Number: 8

Abstract

Abstract The synthesis of a series of benzo (iso) quinoline and phenanthroline derivatives has been achieved using an efficient one-pot procedure. It proceeds through a Suzuki– Miyaura cross-coupling followed by a Dieckmann–Thorpe ring closure under microwave irradiation and provides easy access to building blocks not readily available through other methods.