Improved P1/P1'substituents for cyclic urea based HIV-1 protease inhibitors: synthesis, structure-activity relationship, and X-ray crystal structure analysis

DA Nugiel, K Jacobs, L Cornelius…

Index: Journal of Medicinal Chemistry, , vol. 40, # 10 p. 1465 - 1474

Full Text: HTML

Citation Number: 37

Abstract

... Journal of Medicinal Chemistry. ... The DuPont Merck Pharmaceutical Company, PO Box 80500, Wilmington, Delaware 19880-0500. J. Med. Chem. , 1997, 40 (10), pp 1465–1474. DOI: 10.1021/jm960839i. Publication ...

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