Synthesis and in vitro biological evaluation of mannose-containing prodrugs derived from clinically used HIV-protease inhibitors with improved transepithelial …

…, J Greiner, AM Aubertin, P Vierling

Index: Bashyal, Bharat P.; Fleet, George W. J.; Gough, Max J.; Smith, Paul W. Tetrahedron, 1987 , vol. 43, # 13 p. 3083 - 3094

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Citation Number: 7

Abstract

... Volume: Page ... 3-dimethylaminopropyl)-3-ethyl-carbodiimide hydrochloride (EDC), 4-dimethylaminopyridine (DMAP), lithium hydroxide, pyridine, triethylamine, p-toluenesulfonic acid (p-TsOH), and ... 3.38 (s, 3 H, OCH 3 ), 3.31 (t, J 6.1 Hz, 2 H, H-5), 2.07 (t, J 7.3, 2 ...