e.g. Filippa Pettersson or Cancer Res. 75(6) , 1102-12, (2015) or 10.1002/anie.201600521
Discovery, synthesis, and structure–activity relationship of 6-aminomethyl-7, 8-dihydronaphthalenes as human melanin-concentrating hormone receptor 1 antagonists
M Kamata, T Yamashita, T Imaeda, T Tanaka…
Index: Bioorganic and Medicinal Chemistry, , vol. 19, # 18 p. 5539 - 5552
... Bioorganic & Medicinal Chemistry. ... Pharmaceutical Research Division, Takeda Pharmaceutical Company Limited ... 17 In the present report, we describe the details of our initial medicinal chemistry efforts starting from 1a, focusing especially on a distal phenyl ring, a core scaffold ...