1, 3-Disubstituted benzazepines as neuropeptide Y Y1 receptor antagonists

Y Murakami, S Hagishita, T Okada, M Kii…

Index: Bioorganic and Medicinal Chemistry, , vol. 7, # 8 p. 1703 - 1714

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Citation Number: 11

Abstract

... Bioorganic & Medicinal Chemistry. Volume 7, Issue 8, August 1999, Pages 1703–1714. ... Chemical modifications of 9 gave a potent NPY Y1 antagonist 3-(N-(4-hydroxyphenyl)-N′-methylguanidino)- 1-N-(3-(N′-(tert-butoxycarbonyl)amino)benzyl)-2,3,4,5-tetrahydro-1H-1 ...