Tetrahedron letters

A new versatile linker for the solid-phase synthesis of secondary amines

H Glatz, W Bannwarth

Index: Glatz, Heiko; Bannwarth, Willi Tetrahedron Letters, 2003 , vol. 44, # 1 p. 149 - 152

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Citation Number: 14

Abstract

A novel linker for the solid-phase synthesis of secondary amines based on an intramolecular cyclization was developed. The linker allows for a stepwise built-up of the secondary amines on the support. The feasibility was demonstrated in the parallel synthesis of a small set of different secondary amines.