Synthesis, CoMFA analysis, and receptor docking of 3, 5-diacyl-2, 4-dialkylpyridine derivatives as selective A3 adenosine receptor antagonists

AH Li, S Moro, N Forsyth, N Melman, X Ji…

Index: Journal of Medicinal Chemistry, , vol. 42, # 4 p. 706 - 721

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Citation Number: 201

Abstract

... Journal of Medicinal Chemistry. ... Molecular Recognition Section, Laboratory of Bioorganic Chemistry, National Institute of Diabetes, Digestive and Kidney Diseases, National Institutes of Health, Bethesda, Maryland 20892-0810. J. Med. Chem. ...