e.g. Filippa Pettersson or Cancer Res. 75(6) , 1102-12, (2015) or 10.1002/anie.201600521
Tetrahedron Letters
Synthesis of 2-bromo-7-methyl-3, 5-dihydro-imidazo [4, 5-d] pyridazin-4-one and 3-alkyl-2-bromo-3, 5-dihydro-imidazo [4, 5-d] pyridazin-4-one and their selective …
Two synthetic routes to the versatile 3, 5-dihydro-imidazo [4, 5-d] pyridazin-4-ones 2 and 5 have been developed that allow the production of multigram quantities without the need of any chromatographic purification. Broad and selective elaboration of the heteroaromatic scaffolds has also been accomplished.