e.g. Filippa Pettersson or Cancer Res. 75(6) , 1102-12, (2015) or 10.1002/anie.201600521
Synthesis of novel GABA uptake inhibitors. 4. 1 Bioisosteric transformation and successive optimization of known GABA uptake inhibitors leading to a series of potent …
KE Andersen, JL Sørensen, PO Huusfeldt…
Index: Journal of Medicinal Chemistry, , vol. 42, # 21 p. 4281 - 4291
... Journal of Medicinal Chemistry. ... Chemistry. The overall general strategy used for the preparation of the new compounds presented in Table 1 was via N-alkylation of the parent cyclic amino acids 1 or 2, 46 with the appropriate ...