Synthesis, topoisomerase I inhibitory activity, and in vivo evaluation of 11-azacamptothecin analogs

DE Uehling, SS Nanthakumar, D Croom…

Index: Journal of Medicinal Chemistry, , vol. 38, # 7 p. 1106 - 1118

Full Text: HTML

Citation Number: 50

Abstract

... 0022-2623/95/1838-1106$09.00/0 0 1995 American Chemical Society Page 2. 11- Azacamptothecin Analogs Chart 1 ... Page 5. 1110 Journal of Medicinal Chemistry, 1995, Vol. 38, No. 7 Table 1. ll-Aza-(20S)-camptothecin N-Oxides or N-(Methyl iodide) Salts R ...