Molecules

Bohlmann-Rahtz Cyclodehydration of Aminodienones to Pyridines Using N-Iodosuccinimide

MC Bagley, C Glover

Index: Bagley, Mark C.; Glover, Christian Molecules, 2010 , vol. 15, # 5 p. 3211 - 3227

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Citation Number: 9

Abstract

Abstract Cyclodehydration of Bohlmann-Rahtz aminodienone intermediates using N- iodosuccinimide as a Lewis acid proceeds at low temperature under very mild conditions to give the corresponding 2, 3, 6-trisubstituted pyridines in high yield and with total regiocontrol. Keywords:

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