[3 H]-(R)-NPTS, a radioligand for the type 1 glycine transporter

…, K Fisher, C Strick, L Lebel, C Schmidt, D Hiller…

Index: Lowe 3rd., John A; Drozda, Susan E; Fisher, Katherine; Strick, Christine; Lebel, Lorraine; Schmidt, Christopher; Hiller, Donna; Zandi, Kathleen S Bioorganic and medicinal chemistry letters, 2003 , vol. 13, # 7 p. 1291 - 1292

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Citation Number: 26

Abstract

Download PDF Opens in a new window. Article suggestions will be shown in a dialog on return to ScienceDirect. ... Please enable JavaScript to use all the features on this page. ... The synthesis of NPTS, 6, a potent inhibitor of the type 1 glycine transporter (GlyT1) is described, as well as preparation of 6 in optically active and tritiated form for use as a radioligand for affinity displacement assay of GlyT1. ... The synthesis of NPTS, 6, a potent inhibitor of the type 1 glycine ...